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۽ѧҽҩѧԺԺ潲ѧ

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۴ѧҽѧԺڷϴ˱ҷ٣ѧǰͬһͼ
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ڿ: Journal of Ethno-Pharmacology 2005; 99: 61-67
Ŀ: Influence of co-administrated sinomenine on pharmacokinetic 
fate of paeoniflorin in unrestrained conscious rats.
ͨѶߣ½Ȫ
ߣܻ־ꡢYuen-Fan WongYing Xieۡ
ϲ (ҽо)
Ͷʱ: 2004810
ʱ: 20055 (Available online: 2005320)
http://wlv.openrepository.com/wlv/bitstream/2436/9847/1/Kelvin+Chan4.pdf
1 (Corrigendum)
ʱ: 2007123
http://www.aapspharmaceutica.com/search/view.asp?ID=92993
 
2
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Ŀ: The pharmacokinetics and tissue distribution of sinomenine 
in rats and its protein binding ability in vitro.
ͨѶߣ
ߣ½Ȫܻ־ꡢYuen-Fan Wongϲ (
ҽо)
Ͷʱ: 200521
ʱ: 2005114
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2 (Corrigendum)
ʱ: 2008220
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3
ڿ: Journal of Pharmacological Sciences 2005; 99: 381-391
Ŀ: Pharmacokinetic interaction of paeoniflorin and sinomenine: 
Pharmacokinetic parameters and tissue distribution characteristics in 
rats and protein binding ability in vitro.
ͨѶߣ
ߣ־ꡢ½ȪܻYuen-Fan Wong顢ϲ 
(ҽо)
Ͷʱ: 2005812
ʱ: 200512
http://www.jstage.jst.go.jp/article/jphs/99/4/99_381/_article
3 (Erratum)
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ʵҽӦ֮Чôҽͱȷط֮Ч
һ۶ֻʷ˶ſԱܣΪʲôΪҽҩƵ
ƷΧѾЧִҽѧƳ棬ЩƳ涼Чģʹ
ԼЧҲǾоȷܸЧķʹ
κоʹЧԸ㲻ķڿѧ󳫵Ľ
ǲԱܵġ

ҽҽҩҵľأ뽡һ
⣬ҽҽš񺺡Լڽ̣йĦ˵
ھҪΪһṩ֮ȡá
ĿѧչҽѾǺʵȡѹԵλΪһ
޿ӵߣľ߶֮ɥʧԽ뼲ķʸһ
ҽһҵͶҽļź̶ܴȵΣΪ㴦ҽ
ҵҵΣôͶҵӵҳάYou 
owe it to the PROFESSIONÿһҽڽҽҵ֮Ƿ
ҵĻرҽƻбҵĻרҵˮ׼
άҵ棬طҵߡķԴžԵ
ЧʱַԼҵΣҲΡ

ҽҽҩ̬ȼǶҽҵıѣҲǶὫҽ
ޱؽҽεıѣҲǶṫıѡһͨ
˿ԶҽҩɣΪѭߵ·ҵҽѧȨѰרҵ
нһưȷѡ񣬶ҽûУҽľ
ǽռˣ޻ͷ֮·ҽҽҩֱ̬
ȣ˵Ҳֱ֪ӵòһԣǿɳܵģΪҽ
ǵְ𡪡ΪĿߡ

̷ҲҽһԹйҽᾭõλͣ޲
ĽҽܵľλѵûҪȡ
ӦᾭõλҪԼȥYou have to EARN itôȥ
ʰһԼɵ椵԰ա

ʹߣйҽҲһ˼άʵաˣ
ҽѧʦϣףһԼܶ˵ʲôҸҵ˳裬
Ҹҵ˽Ľ̵ҡСġ
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йҽձҪǿԼרҵ

(XYS20080403)

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ֻҪгãйҽעʧܡذ̷

Ѱ

ϲ飬һϴүҪղ߹ſڵһ꼶
ѧ֪ܲҪ̽ƣͣͷʮ㡣
ҽԱĵòһ̸ҽģ˶кܶ


йҽѰʼ˿ʱȳ˺ܾˣ
˸˲ҩйҽĴ˫
̥İ̥ڶʮ̥ˣмBֲ״ÿһ
̥Ѳ̶ȼӱйҽģҲѣвס

ҶйҽģҽĺȤضԣֻҪ
ҽɳ֪ǵġѧߡذɡеҽķУ
ܿľ;ԣֻ֯ķץסʵʣйҪ
ǡƽЧ桢֯ķտֻĽ
֣Ϊû˶𣬿ЩΧǵЩ뵱Ȼġרҡ
Ҳࡣ

йռ񾭼õ5.5%ΧʵȫҽƱĹȲ
ͣҲ˵ڹ񾭼еռԵģ
ռʸߣôҽƷõȷߣڹҺϵδأ֧ߣ
ҲߣôľҵְλҲࡣϵΨһָ
Ч棬Ҫѧٵľѧѧ˷ú֪˻Ƚϳ
Ӧ֪ӻƻ󣨵Ȼ۸ˣҪһ֪

й˵ӦøȫҽȱйҪꡢʮꡢ
ʮһȡй̶ȣȡ
ҽг̶ȡйȫҽйҽϵӵز
йϵܰŶˣǼӴƾͲˡȫҽ
ζֱӿȼӴ󣬳˵ٵģ˭ûкùӳԡ

йҽϵ˵˾ظߵĹɱɱֳ࣬
ϤĸֻռС֣󲿷޴뵱ȻɵģҲǷȱƣ
йһ棬ǲ˵ģеĵͼƽ⣬йȱȽǡй
뾭һг̣ʹгЧ棬йҲһ
гһп˼롢ںҽƴҵԱйǰƻ
õʧܾǹʤĳԵʧܣֱ죬йҽԱ
ȻΪ֮򵥣йҽƽԱҪѧԼԣ
Ҫһܲվյͷ

йҽ䲻ҪϣһΰҽķԺܿıǵ
йǰηΧƶ²ҽ⣬
ƵԱһȱʵʹ飬ȱԶĿ꣬ƾ뵱Ȼ飬
ҽԱ˵õķάҽԱˮƽķõķ
ͺ˵ˡҽԱ߳һµģʶ
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йеҽͻǻҽԱṩķδܲ
ҽƺģʵϾҽԺշѻϲ
ҽףҽԺǮһˣ߶ʵúܡйѧĹʽҽƣ
ĳЩᵽͷѡ൱ҵİϣеҽϵ
ص͹ҽԺɱγɵĸѱ׼ػ½
ʱйɸˡ

˿ϿչڶйҽʧúܣȻйĸ
ûҽϲУйҽĶѾҶǵ
κϣˡ̷йǮҵϺǹģԶ
60ҽƸĸʱǮ࣬ҽǷԡ
йҽⲻͶ⣬Ͷ࣬йִҵ
ΪֹҽҵһֺֻܰԵһëǮҪ
һԪǮйҽüͷдְƣǲʵ֣
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йҽƵһѼͥ⣬ǸĸеĹ
ҽԺŮʲôأŮûж̣ĸæΪŮι̡ϴ
򲼡ƨɣûлͣһԼŮδŮأ
Զ󣬹˶ڵˮûӪûԾ͵ðĸʲô
뵽ˣŮͺȤѧϰҲûн
һǵļͥ

йҽΣһ⣬⣬Ҳҽ⣬
ߵ⡣Ҫ׼ԼλãҽҲҪԼľҲ
Ŭϵˣ϶ϵ÷ɲˣδغóԡ
ĸйҽΣ롣ΪʲôѰйȳ
ĸ鰸Ȥԭ

Ȥĸĸ¶ϵĸĸ˭⣬˭ͽԼ⣬
ֱ⣬Ҫϵʱٷ߸ĸˮ
ɣһõĽ飬Ǿˮ£˵ԶȴҲţ
й۲ʲôƣҽҽʿĻʿ
ԱĹԱйҽΣֻиơ

йҽҵҪıǾҲѧ֯ţ
ƽЧ桢йȻӡˢƱǾζԴ
ǮȽȵ˵Ǯɱڵ
һðյ顣

ѰûȤĹ٣ҲûȤһʲôҩʽķ
ҡҴæݽίİͷϡҿйгǧ
ίǸֵȤĹҲλͲı
Բò̷ʽҽʧˣ뷢ί֮
£ҽһζһҽ

ãûѳԺʿߣҽҲҽߣ
ùǲġѰûиĸйҽϵһӼƻʹУҲ
õԺǰȥְȨ档˿ϵĶߣ
ؽԼ˼·й⡪ǾģҴӲ
ΪԼĹ۵㵣

˵һݹһ棬ԼƨԼйĲҽ
ѰΪҪʰԼ⣬еԼΡ

һƪ˼·̫ȷҲ˰̷ġ

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㶫ѧʦѧλ

:!

ѧٵĴ,ֵ½˿վ,ебҪһ
ɵѧٽҷ,֪Ϸ,ֻ.

һżȻϿУʦľȻǻϲ,
رȫϮ,ʵǻƵ˼.

1ƪɵġ½ṹɿԹӦо(ɽƼѧ
ʿ),һƪԬչ˶ʿѧλġ۹ṹĿɿԷ(пƼ
ѧ˶ʿ) .ǰߵĸûֵ,ڳϮƴվȲ,ƪ
ݲһ,һ,ֱ˼.һѧԺ,ͬʱ
ᵽлǰߵİ.ְʵڱ.

㶫ѧһʦ

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Ϊ˺ʵһʵй֪ݿԡаС
ۡΪҽڡڿݿ⡱вѯһ75ƪ£
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ģҴԼһ75ƪУ뻯ѧֱص51ƪ
йػԵ⣨ѧĿȣҵĸ£

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ʱ䣬ȤĻҷЩйسѧġ
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2۲ʶֻǸоڻСѧڵ
Що顣ֻΪ׬ЩѣҲְ
ҪȻѧۡ

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ڿлĽ

laoma

һõĿлӦùͶıȽϡĿǷȷ
ʵδﵽĿķж󣬵ͶǷ

ڵһʱûкð취ﳢۺ⡣

ڶǡշίĻӦƫСյģƼĿ
Գܸ߷յĿⲢ˵ǮϹӡڷԤͨõֶǽ
ģͣʷơӵģкܶҪ
ûкܺõģ֮ǰԲȫʷһӴĲԡ

ᵽ⣬֪ĳ˵ǰļ¼ʱԸ
۵ǳȷҲǿġͰԱȼ뵥λ
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ҵзոߵĳԡһǿĿϢϵͳ
˶κεطκʱٲѯκ˵ü¼ò
罻׵ãǻˣ뵥λ˵á

ʷԽ࣬ԽķԤ׼ȷزǰӦ
û˺ܶԼʷݣרҿ⣬ǰĿյĲϵȡ
һϢϵͳһǰûĿˣϵͳ
ڶξҪѡпһŵľѡ˵
ǿĿϢϵͳӦзֲڸءŵݿĲѯܡɰ
˵Ŀʷ¼Ͷʷоɹרҵʷ¼
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Ŀȵȡ

ITϻܴѡITҪͳһ
ݽʽݿͻ©Ƚи죬ԣӦȵȡ
ܴ󣬷ÿڣʵʩʱҲܳϵìܻᷢڼ
ЭϣǷԸԼó˭ݸʽΪ
׼ȡӹҽǶȿӦôӸߵĲЭͶϢϵͳʡ
ķúֲܿϵͳͶʣҲ߹ţ֪
ǺúƵġ

ϵͳҲҪƹ㣬һôңˡλѯ
һôҼݡ

ǡͶ롱ָ涨Ŀ¼֧Լ۱ȵ۱
ϸӣ׻˵һǮһֻһëǮֻһǮֻһ
Ŀ趨Уﲻۡ

ĿĿļָ꣬ȻĿǩʱ͵͵
ʱָ꣬Ǹ࿿ϵõĿرר𣬲ûаԴ
ӦĿĿϣ̰ۡ繺ֵϳСؼң
½ѿ˾ǮתȥĻǺټרĿ鳤
𣬵ƣԽ⡣

רĿ鳤Բָʽһ˻Ŀص
֧Ӹ˻Ŀ鳤ǩ֧䡣ʻɵλάί
ϵĻά鳤շѺͷѡ鳤ܲ񣬵
֪Ǯʲôط˻άԶṩĿ鳤
ܶлҪ˴Բ뿴ɣһУԼٸĿ
ȥÿĿ֧

ڻͨסԳҪ󣬶˻ʹǷס
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һڵλͳ̣Ŀ鳤òǮʹĿܰʱɡڱҪʱ
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Ҫʽϱ֤ʽʹõõĿкͽ
Ȼ˶֣˶Թʡɹ÷Ƿͬϵ
һ£ϼʱӷǷöԣƱǲٵģ˲
Ƿһ£˲ͻܱǷԵϡȻ󿴳Ƿԣ籨
ϵǩǲȫɹǰǷңǷб꣬ǷкͬǷִ
кͬǷգƷǷˣߵĹҪǩ֡Ȼ̵㣬
ȻԱ֪豸ǸʲôģǺ˶ʵ˲ϵıţ
ܶ൥λԱڱĵطĶʶġ
ҪΪ覴õĵطҪλṩ˵Ҫʾλ
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Ҫ˵Ϊʲôñˣǲʱ鱨ıʽ;ʽ
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øĴۡǽԼɱһַղǺܱҪġ
ͬʱһĿЭùͬίУֻһ顣

ҪоȵļγɹҪ߼豸
дҪĳ豸ĿɺлҪܶ
ͷһߣʹáĿƵĿҪһ̨
ɺܶ൥λи豸ÿ̨ʹʶߡ

Գһƽ̨߼豸Ŀʱƽ
̨κ˿гʹá豸ڵλӪ򹫹ƽ̨
ʹƽ̨άƹ㣬ôʹø豸ʹЧ
ߵ豸ƽ̨Կۼ۴ҵлҪʹ
ʱԲٹ豸ֻҪʹ÷ѾͿˡ

Ľ鶼ҪǮʡӦñȸĶࡣ˺ˣΣ
ƽ̨ӦԵģȳϢϵͳҪˡ

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ҵҩƷؿ԰

lw56102

ҩƷؿҽмһܣҲùڲҽˣ
ᵱҲáҲΪʲô˵ģ£

һҩƷؿҲãҲ棬ȫҽҩ
һͬѧʼһʱǮһʱΪڿƵˡ
˿ſϣΪЩֹܻؿ۵Ժ쵼ǰûչؿۣ
㲻գõЩҩƷҲήۣ㲻Ҫǲȫҩ

ڶܹΪҩƷؿӰԼĴΪ˵
ҩƷؿԴڸҩҩΪ࣬ӱƼH2׿
ԱˣǰЧáǰڲҪþƼΪĺͽ
ڵģڷҩЧܴ󣬵õЧ൱ҹıȽڵıˣ
лؿۣڵ޻ؿۣɵӶ֪ѡһЩԷѵľ
ĲˣҲһѡӱƼڲ£һ
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ãһθ׻߶ãΪʵҪãѡ
ϳù࣬۸ˣ׽խȻ޻ؿۡ

⼸㣬Ҷߵͬ¹۲죬󲿷ܹġ漰
ҩڲҩҪԾҩΪҲҪʣסԺѵ
Ͳÿڷҩ𣿵Ȼԣڷ׻ߣ̿ҲûнһҪ
ǲסԺ̶ܴϾΪ˴뷽㣬סԺֻڷҩ
߻סԺû塣Ȼ漰йҽסԺ׼յ⣬
ܸӣڱҪֵ̽ݡϣܶҽڲҩ
ƷؿԴﵽһ߳Ҫؾ
˵Ͳ顣ܵĴλһֱԱҶ˲
ΣأôӦҩʱͻ󣬷ĳ²٣
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ȻֻҸˣкܶȽϤͬʵҽҲᡣÿҲ
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ÿµȴȲҪһ롣һΪĲ˴Ƚᣬ
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гҩźܶȥҽԺĶƾҽʦڿƻƣ
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Ʒһ廨ŵгҩгҩļ۸ռܼ۸൱
ɷ֣ҩļ۸ֻгҩ۸һͷ

ҽԺгҩҽ֮һǴζŴ
ӴӴҽҩһҴгҩŵĻؿ
ԼҩƷ۸10%-20%֮䡣Ҷгҩ̬ȴ¾˲
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ݣҲԲˡֺܶгҩӦ֢Ӧ
ٴҲȱгҩĲӦý屨У
ҲСйҽǻҽûϱҩﲻӦϰߣ
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ˣʱ͵һʱ䡣

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ԪǿƵӶ

ׯ

42գ̨˴Ԫרǡǿר
Ƭ̸ҽϵ

ǿڽĿ˵ڵҽ飬ҽһÿ궼һ
ҽģǲӦùעţӦùעš

˶ۣЦԷǡ

ÿ궼һҽģǸʲôǲȫ
ʡսʮģй֮󣬾ȱиҽµİ
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ҽԺȫƷһסԺƣͬ˲ӵŰס
ҩ߼ۼ顢߼۷ȫԺ˵㡣ͨͥһ˻˴󲡣
˲աҽԺͨǲ۲۵ϵ۶صĲ飬
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ԸǶ֮ȡҽԺ˸ţǻƲƣǻ
ߺ׼ܲνţԺǮ
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Ҷ֪ľͰۡľͰʢˮٵĲľ
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ҽߡý͹ֻнסЩĲ֣٣ʹ֮
ĽſʵˮǴߡǿǹȻԲѵôҲľ
жӵĳľⲻǵ͵Ķ

ǿⷬر204ҽߵǣ
Ǳ13ڹ˽ǡ

ʵǿԪĶԻǸѥɦ˭֪ҽϵ
ĸԭ˰˶Թ֧ûзȨලȨȨų
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ⲻǿԪƸҲãҲգǷ곡Ϸ
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Ҫҽ

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˼ˡҽܾе㲻ζҽ
ϡѧרмһˡ㣬Ӧٶ֪ۡ
ʶϻȵȣĸʱ򿴵Ĵֱҽ
ҽʵΪҲǸġҽ
ҵҵһ಻ͬˣҵſԳչʹ
ҽҲҪϡ

һҽҪ飺һҽѧУ飨Ҳμӹ
֪ʶѧϰһٴʵԼľܽᣬϼҽ
ڵľܽᡣǰһǱ˵ľ飬һԼľ(һ
ʦб˵ľ)ֻǰһûжǱҽ
é®ҽֻڹвܽʵ飨ɹʧܣ
ʹһ齥β˲Ųңٳ͵Ӧ֡
β˵ҽǾûеġ

ٴҽѧʦйϵǺҪġʦͽҵˡֻ
׷ԲԵҽѿ˵ĲƸǰҽڹ
пҽѿĲҽ̡һҽӦ
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õķ˵ʹ࣬˵һЩΪǵ˶ʿʿҽ
Ų¼оҽʿǲʧȥΪ
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ΪáèۡжҽòýΪʵʣǣҽۣ
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